Pharmacological Comparative Characterization of REL-1017 (Esmethadone-HCl) and Other NMDAR Channel Blockers in Human Heterodimeric N-Methyl-D-Aspartate Receptors

Sabato 13 agosto 2022 circa 1 minuti di lettura

Journal and Affiliations:

Pharmaceuticals, 13 agosto 2022

Jacopo Sgrignani, Istituto di Ricerca in Biomedicina, Bellinzona

Patrizia Locatelli, Istituto di Ricerca in Biomedicina, Bellinzona

Andrea Cavalli, Istituto di Ricerca in Biomedicina, Bellinzona

Andrea Alimonti, Istituto oncologico di ricerca, Università della Svizzera italiana, Bellinzona

Tags:
d-methadone
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dextromethadone
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dextromethorphan
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esmethadone HCL
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ketamine
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major depressive disorder (MDD)
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memantine
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MK-801
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N-methyl-D-aspartate receptor (NMDAR)
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REL-1017
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Authors:

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Andrea Alimonti
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Andrea Cavalli
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Jacopo Sgrignani
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Patrizia Locatelli
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Link: https://www.mdpi.com/1424-8247/15/8/997&